A = almost entirely absorbed, 25% reaches systemic circulation via liver metabolism. peak plasma conc. 1-4 hours after administration. Bioavailability increases by up to 50% with food consumption
D = vol. - 4L/kg, 90% plasma protein bound (albumin)
5 of 6
Propranolol:
Metabolism? Elimination?
M = high 1st pass by liver. 42% aromatic hydroxylation, 41% N-dealkylation -> side chain oxidation, 17% direct glucuronidation (individual variants)
E = majority via urine
6 of 6
Other cards in this set
Card 2
Front
Propranolol:
Indications? Cautions?
Back
I = Thyrotoxicosis, Hypertension, Anxiety
C = Bronchospasm, hypotension, psoriasis
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